Oxygen

Class Vital ingredient of multicellular life
Chemistry

Diatomic gas

Routes of administration

Inhaled; also as intravenous or intra-arterial infusion of well-oxygenated blood (i.e. ECMO), and can be given externally (as in hyperbaric oxygen therapy)

Absorption

Absorbs rapidly into the pulmonary circulation via the lungs (250ml/min with 21% FiO2, at rest)

Solubility

Poor solubility in water

Distribution

Widely distributed- total body oxygen content is 64% by weight. Highly protein-bound (to haemoglobin)

Metabolism

Metabolised in all tissues (mainly brain, heart and skeletal muscle)
Mainly metabolised by cytochrome c mitochondrial enzymes (90%)
Zero-order clearance kinetics, roughly 200ml/minute

Elimination

Rapidly eliminated by metabolism into CO2 and water

Time course of action

Minutes

Target receptor

Cytochrome c mitochondrial enzymes

Mechanism of action

Increases ATP by acting a substrate for aerobic metabolism of glucose

Clinical effects

Drying of mucous membranes and inspissation of secretions

Inflammatory tracheobronchitis

Decreased central respiratory drive (minimally)

Hypecapnoea in "CO2 retainers" mainly by virtue of V/Q mismatch and Haldane effect

\Absorption atelectasis Increased left-to-right shunting in ASDs

Increased peripheral vascular resistance

Cerebral and coronary vasoconstriction

Euphoria

Retrolental fibroplasia of the newborn

Decreased erythropoiesis

Literature reference

Haim Bitterman's 2009 article, "Bench-to-bedside review: oxygen as a drug"

CICM details of understanding Level 1
Mentioned around Deranged Physiology
Related SAQs

Question 1 from the first paper of 2011

Question 6 from the first paper of 2009

Question 14 from the first paper of 2023